Research Use Only - Not for human consumption. 18+ only.
Research CompoundKhavinson BioregulatorsSubcutaneousOral

Pinealon

Also known as: EDR tripeptide, Brain bioregulator

Pinealon is a Khavinson bioregulator for the brain and nervous system. It consists of three amino acids (Glu-Asp-Arg) and supports cognitive function and neuroprotection.

Research Status

Research Compound

Research compound

For research purposes only. Not approved for human use. Not medical advice.

Research Areas

Neuroprotective effects
Improves memory and learning
Supports brain health
May reduce cognitive decline
Regulates circadian rhythm
Anti-aging for the brain

Side Effects

Injection site reactions
UncommonMild

Minor redness, swelling, or itching at the injection site may occur. Rotate injection sites to minimize this risk. Reactions typically resolve within 24 hours.

Sleep disturbance (initial)
UncommonMild

Some users report vivid dreams or mild insomnia during the first few days of use, likely due to enhanced melatonin signaling. This typically resolves as the body adapts. Consider injecting in the morning rather than evening.

Headache
RareMild

Occasional mild headache has been reported in early treatment phases. Ensure adequate hydration and consider timing of injection relative to meals.

Dizziness or lightheadedness
RareMild

Rare reports of transient dizziness. Sit or lie down for a few minutes after injection if this occurs. Discontinue and consult a healthcare provider if symptoms persist.

Allergic reaction
RareSerious

Although rare, allergic reactions (rash, urticaria, difficulty breathing, angioedema) are possible with any peptide. Seek immediate medical attention if signs of anaphylaxis occur. Discontinue use and do not re-administer.

Dosing Reference

ParameterValue
Dose range10 mg
FrequencyDaily for 10-20 days per month
TimingMorning
RouteSubcutaneous, Oral

Cycle 10-20 days on, 10+ days off. Part of bioregulator family.

Research disclaimer

Figures drawn from published research literature and community logs. Not clinical recommendations. Consult a qualified professional. Research use only.

Reconstitution Guide

Do not use saline or bacteriostatic saline — use only bacteriostatic water for reconstitution

Do not shake the vial vigorously; gentle swirling prevents peptide degradation

Discard immediately if the solution appears cloudy, discolored, or contains visible particles

Use within 30 days of reconstitution when stored at 2–8°C

Do not freeze the reconstituted solution; freezing may denature the peptide

Use the PeptideVolt reconstitution calculator for your exact concentration

Use the PeptideVolt reconstitution calculator for your exact concentration

Molecular and Pharmacological Data

SequenceGlu-Asp-Arg

Pinealon (Glu-Asp-Arg) is a Khavinson bioregulator tripeptide that supports pineal gland function and neuroprotection through regulation of melatonin synthesis and circadian rhythm stabilization. It is believed to enhance cognitive function, improve sleep quality, and provide antioxidant protection to the central nervous system by modulating neuroendocrine signaling and reducing oxidative stress in brain tissue.

Pineal Gland Regulation

Pinealon is hypothesized to support pineal gland function and melatonin production, which regulates circadian rhythms and sleep-wake cycles. Enhanced melatonin signaling may improve sleep quality and cognitive performance.

Neuroprotection and Antioxidant Defense

The tripeptide composition (glutamic acid, aspartic acid, arginine) may provide antioxidant and neuroprotective effects, reducing oxidative stress and supporting neuronal survival in aging or stressed neural tissue.

Neuroendocrine Signaling

Bioregulator peptides are thought to modulate neuroendocrine communication, supporting healthy aging of the nervous system and maintaining cognitive reserve.

  • Pinealon is part of the Khavinson bioregulator family, a class of short peptides derived from animal tissues designed to support organ-specific function
  • The tripeptide sequence (three amino acids) is small enough for potential oral absorption, though subcutaneous injection ensures reliable bioavailability
  • Pinealon is typically used in cyclic protocols (10-20 days on, 10+ days off) to maintain responsiveness and avoid tolerance
  • Research on Khavinson bioregulators is primarily published in Russian and Eastern European literature; Western clinical trials are limited

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Research Use Only. All content on this page is provided for informational and educational purposes related to scientific research. Pinealon is not approved for human use by the FDA or any equivalent regulatory body. This is not medical advice. Do not use any substance discussed here for therapeutic, diagnostic, or preventative purposes. Consult a qualified healthcare professional before making any health-related decisions. The Peptide Volt does not endorse the use of any research chemicals. 18+ only.