Research Use Only - Not for human consumption. 18+ only.
CGrade CPrimarily animal or in-vitro studies; limited human dataResearch OnlyResearch OnlyNo regulatory approval in any major jurisdiction; for research use onlySkin & Anti-AgingSubcutaneous

Pentapeptide-18

A synthetic pentapeptide that inhibits acetylcholine release at the neuromuscular junction, reducing facial muscle contractions and wrinkle formation.

Research Status

CGrade CPrimarily animal or in-vitro studies; limited human dataResearch OnlyResearch OnlyNo regulatory approval in any major jurisdiction; for research use only

Research compound

For research purposes only. Not approved for human use. Not medical advice.

Research Areas

Reduces facial muscle contractions and wrinkle formation
Inhibits acetylcholine release at neuromuscular junction
Potential anti-aging effects on skin appearance
May improve skin texture and elasticity
Research compound for cosmetic applications

Side Effects

Skin irritation or redness
UncommonMild

May occur with sensitive skin or if applied to compromised skin barrier. Discontinue use if irritation persists beyond 48 hours and consult a dermatologist.

Localized dryness
UncommonMild

Can be managed by applying a non-comedogenic moisturizer after the peptide solution has fully absorbed.

Allergic contact dermatitis
RareModerate

Possible in individuals with peptide sensitivities. Perform a patch test on a small area before full facial application. Discontinue if rash, swelling, or itching develops.

Photosensitivity
RareMild

Some users may experience increased sun sensitivity. Use broad-spectrum SPF 30+ sunscreen during research application periods.

Temporary stinging or tingling
UncommonMild

May occur immediately after application, particularly on sensitive areas around the eyes. Effect typically resolves within minutes.

Dosing Reference

ParameterValue
Dose range5-10 mcg
Frequency, timing and route - members only

Research disclaimer

Figures drawn from published research literature and community logs. Not clinical recommendations. Consult a qualified professional. Research use only.

Reconstitution Guide

Do not use saline or bacteriostatic saline, use only bacteriostatic water for reconstitution

Do not shake the vial vigorously; gentle swirling prevents peptide degradation

Discard immediately if the solution appears cloudy, discolored, or contains visible particles

Use within 30 days of reconstitution when stored at 2-8°C

Do not freeze the reconstituted solution; freezing may denature the peptide

Use the PeptideVolt reconstitution calculator for your exact concentration

Use the PeptideVolt reconstitution calculator for your exact concentration

Molecular and Pharmacological Data

Pentapeptide-18 is a synthetic peptide designed to mimic the inhibitory effects of botulinum toxin by reducing acetylcholine release at the neuromuscular junction. This mechanism decreases facial muscle contractions responsible for dynamic wrinkle formation, particularly in the upper face. The peptide works through a non-toxic pathway to achieve similar cosmetic anti-aging effects.

Pathways and mechanism detail available to members

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Recent Research

All results

Source: PubMed / NCBI. Updated daily. Articles are listed for research reference only.

Research Citations

4 sources
  • Blanes-Mira C, Clemente C, Jodas G, et al. (2002). A synthetic hexapeptide (Argireline) with anti-wrinkle activity. International Journal of Tissue Reactions. 24(4):139-48.

  • Gupta AK, Gover MD. (2006). Topical peptides and proteins in dermatology. American Journal of Clinical Dermatology. 7(2):81-95.

  • PubMed PMID: 12472620 - Study demonstrating acetylcholine inhibition mechanism in synthetic peptides for wrinkle reduction

  • Seiberg M, Paine C, Sharlow E, et al. (2000). The protease-activated receptor 2 is induced in keratinocytes during wound healing. Experimental Dermatology. 9(3):221-228.

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Research Use Only. All content on this page is provided for informational and educational purposes related to scientific research. Pentapeptide-18 is not approved for human use by the FDA or any equivalent regulatory body. This is not medical advice. Do not use any substance discussed here for therapeutic, diagnostic, or preventative purposes. Consult a qualified healthcare professional before making any health-related decisions. The Peptide Volt does not endorse the use of any research chemicals. 18+ only.